Titanium-mediated reductive cross-coupling reactions of imines with terminal alkynes: An efficient route for the synthesis of stereodefined allylic amines
Author(s): Kebin Mao | Guoqin Fan | Yuanhong Liu | Shi Li | Xu You | Dan Liu
Volume: 9
Issue: 1
Year: 2013




N-Heterocyclic carbene–palladium catalysts for the direct arylation of pyrrole derivatives with aryl chlorides
Author(s): Ismail Özdemir | Nevin Gürbüz | Nazan Kaloğlu | Öznur Doğan | Murat Kaloğlu | Christian Bruneau | Henri Doucet
Volume: 9
Issue: 1
Year: 2013




Inclusion of the insecticide fenitrothion in dimethylated-β-cyclodextrin: unusual guest disorder in the solid state and efficient retardation of the hydrolysis rate of the complexed guest in alkaline solution
Author(s): Dyanne L. Cruickshank | Natalia M. Rougier | Raquel V. Vico | Susan A. Bourne | Elba I. Buján | Mino R. Caira | Rita H. de Rossi
Volume: 9
Issue: 1
Year: 2013




Peptoids and polyamines going sweet: Modular synthesis of glycosylated peptoids and polyamines using click chemistry
Author(s): Daniel Fürniss | Timo Mack | Frank Hahn | Sidonie B. L. Vollrath | Katarzyna Koroniak | Ute Schepers | Stefan Bräse
Volume: 9
Issue: 1
Year: 2013




Microwave-assisted three-component domino reaction: Synthesis of indolodiazepinotriazoles
Author(s): Rajesh K. Arigela | Sudhir K. Sharma | Brijesh Kumar | Bijoy Kundu
Volume: 9
Issue: 1
Year: 2013




A new synthetic protocol for coumarin amino acid
Author(s): Xinyi Xu | Xiaosong Hu | Jiangyun Wang
Volume: 9
Issue: 1
Year: 2013




Alkyne hydroarylation with Au N-heterocyclic carbene catalysts
Author(s): Cristina Tubaro | Marco Baron | Andrea Biffis | Marino Basato
Volume: 9
Issue: 1
Year: 2013




Chemical–biological characterization of a cruzain inhibitor reveals a second target and a mammalian off-target
Author(s): Jonathan W. Choy | Clifford Bryant | Claudia M. Calvet | Patricia S. Doyle | Shamila S. Gunatilleke | Siegfried S. F. Leung | Kenny K. H. Ang | Steven Chen | Jiri Gut | Juan A. Oses-Prieto | Jonathan B. Johnston | Michelle R. Arkin | Alma L. Burlingame | Jack Taunton | Matthew P. Jacobson | James M. McKerrow | Larissa M. Podust | Adam R. Renslo
Volume: 9
Issue: 1
Year: 2013




Facile synthesis of benzothiadiazine 1,1-dioxides, a precursor of RSV inhibitors, by tandem amidation/intramolecular aza-Wittig reaction
Author(s): Krishna C. Majumdar | Sintu Ganai
Volume: 9
Issue: 1
Year: 2013




Asymmetric Diels–Alder reaction with >C=P– functionality of the 2-phosphaindolizine-η1-P-aluminium(O-menthoxy) dichloride complex: experimental and theoretical results
Author(s): Rajendra K. Jangid | Nidhi Sogani | Neelima Gupta | Raj K. Bansal | Moritz von Hopffgarten | Gernot Frenking
Volume: 9
Issue: 1
Year: 2013




Complete σ* intramolecular aromatic hydroxylation mechanism through O2 activation by a Schiff base macrocyclic dicopper(I) complex
Author(s): Albert Poater | Miquel Solà
Volume: 9
Issue: 1
Year: 2013




Zanthoxoaporphines A–C: Three new larvicidal dibenzo[de,g]quinolin-7-one alkaloids from Zanthoxylum paracanthum (Rutaceae)
Author(s): Fidelis N. Samita | Louis P. Sandjo | Isaiah O. Ndiege | Ahmed Hassanali | Wilber Lwande
Volume: 9
Issue: 1
Year: 2013




Development of peptidomimetic ligands of Pro-Leu-Gly-NH2 as allosteric modulators of the dopamine D2 receptor
Author(s): Swapna Bhagwanth | Ram K. Mishra | Rodney L. Johnson
Volume: 9
Issue: 1
Year: 2013




A new synthetic access to 2-N-(glycosyl)thiosemicarbazides from 3-N-(glycosyl)oxadiazolinethiones and the regioselectivity of the glycosylation of their oxadiazolinethione precursors
Author(s): El Sayed H. El Ashry | El Sayed H. El Tamany | Mohy El Din Abdel Fattah | Mohamed R. E. Aly | Ahmed T. A. Boraei | Axel Duerkop
Volume: 9
Issue: 1
Year: 2013




Amino-substituted diazocines as pincer-type photochromic switches
Author(s): Hanno Sell | Christian Näther | Rainer Herges
Volume: 9
Issue: 1
Year: 2013




Synthesis of spiro[dihydropyridine-oxindoles] via three-component reaction of arylamine, isatin and cyclopentane-1,3-dione
Author(s): Yan Sun | Jing Sun | Chao-Guo Yan
Volume: 9
Issue: 1
Year: 2013




Tandem aldehyde–alkyne–amine coupling/cycloisomerization: A new synthesis of coumarins
Author(s): Maddi Sridhar Reddy | Nuligonda Thirupathi | Madala Haribabu
Volume: 9
Issue: 1
Year: 2013




Carbolithiation of N-alkenyl ureas and N-alkenyl carbamates
Author(s): Julien Lefranc | Alberto Minassi | Jonathan Clayden
Volume: 9
Issue: 1
Year: 2013




Enantioselective reduction of ketoimines promoted by easily available (S)-proline derivatives
Author(s): Martina Bonsignore | Maurizio Benaglia | Laura Raimondi | Manuel Orlandi | Giuseppe Celentano
Volume: 9
Issue: 1
Year: 2013




De novo synthesis of D- and L-fucosamine containing disaccharides
Author(s): Daniele Leonori | Peter H. Seeberger
Volume: 9
Issue: 1
Year: 2013




An improved synthesis of a fluorophosphonate–polyethylene glycol–biotin probe and its use against competitive substrates
Author(s): Hao Xu | Hairat Sabit | Gordon L. Amidon | H. D. Hollis Showalter
Volume: 9
Issue: 1
Year: 2013




A one-pot catalyst-free synthesis of functionalized pyrrolo[1,2-a]quinoxaline derivatives from benzene-1,2-diamine, acetylenedicarboxylates and ethyl bromopyruvate
Author(s): Mohammad Piltan | Loghman Moradi | Golaleh Abasi | Seyed Amir Zarei
Volume: 9
Issue: 1
Year: 2013




A peptidic hydrogel that may behave as a “Trojan Horse”
Author(s): Nicola Castellucci | Giorgio Sartor | Natalia Calonghi | Carola Parolin | Giuseppe Falini | Claudia Tomasini
Volume: 9
Issue: 1
Year: 2013




Synthesis and evaluation of cell-permeable biotinylated PU-H71 derivatives as tumor Hsp90 probes
Author(s): Tony Taldone | Anna Rodina | Erica M. DaGama Gomes | Matthew Riolo | Hardik J. Patel | Raul Alonso-Sabadell | Danuta Zatorska | Maulik R. Patel | Sarah Kishinevsky | Gabriela Chiosis
Volume: 9
Issue: 1
Year: 2013




New GABA amides activating GABAA-receptors
Author(s): Peter Raster | Andreas Späth | Svetlana Bultakova | Pau Gorostiza | Burkhard König | Piotr Bregestovski
Volume: 9
Issue: 1
Year: 2013




Alternaric acid: formal synthesis and related studies
Author(s): Michael C. Slade | Jeffrey S. Johnson
Volume: 9
Issue: 1
Year: 2013




Synthesis of SF5-containing benzisoxazoles, quinolines, and quinazolines by the Davis reaction of nitro-(pentafluorosulfanyl)benzenes
Author(s): Petr Beier | Tereza Pastýříková
Volume: 9
Issue: 1
Year: 2013




Thioester derivatives of the natural product psammaplin A as potent histone deacetylase inhibitors
Author(s): Matthias G. J. Baud | Thomas Leiser | Vanessa Petrucci | Mekala Gunaratnam | Stephen Neidle | Franz-Josef Meyer-Almes | Matthew J. Fuchter
Volume: 9
Issue: 1
Year: 2013




Some aspects of radical chemistry in the assembly of complex molecular architectures
Author(s): Béatrice Quiclet-Sire | Samir Z. Zard
Volume: 9
Issue: 1
Year: 2013




A computational study of base-catalyzed reactions of cyclic 1,2-diones: cyclobutane-1,2-dione
Author(s): Nargis Sultana | Walter M. F. Fabian
Volume: 9
Issue: 1
Year: 2013




Iron-containing mesoporous aluminosilicate catalyzed direct alkenylation of phenols: Facile synthesis of 1,1-diarylalkenes
Author(s): Satyajit Haldar | Subratanath Koner
Volume: 9
Issue: 1
Year: 2013




Spin state switching in iron coordination compounds
Author(s): Philipp Gütlich | Ana B. Gaspar | Yann Garcia
Volume: 9
Issue: 1
Year: 2013




Recent advances in transition-metal-catalyzed intermolecular carbomagnesiation and carbozincation
Author(s): Kei Murakami | Hideki Yorimitsu
Volume: 9
Issue: 1
Year: 2013




Synthesis of 5-(ethylsulfonyl)-2-methoxyaniline: An important pharmacological fragment of VEGFR2 and other inhibitors
Author(s): Miroslav Murár | Gabriela Addová | Andrej Boháč
Volume: 9
Issue: 1
Year: 2013




Inter- and intramolecular enantioselective carbolithiation reactions
Author(s): Asier Gómez-SanJuan | Nuria Sotomayor | Esther Lete
Volume: 9
Issue: 1
Year: 2013




Synthesis and testing of the first azobenzene mannobioside as photoswitchable ligand for the bacterial lectin FimH
Author(s): Vijayanand Chandrasekaran | Katharina Kolbe | Femke Beiroth | Thisbe K. Lindhorst
Volume: 9
Issue: 1
Year: 2013




A new intermediate in the Prins reaction
Author(s): Shinichi Yamabe | Takeshi Fukuda | Shoko Yamazaki
Volume: 9
Issue: 1
Year: 2013




Radical zinc-atom-transfer-based carbozincation of haloalkynes with dialkylzincs
Author(s): Fabrice Chemla | Florian Dulong | Franck Ferreira | Alejandro Pérez-Luna
Volume: 9
Issue: 1
Year: 2013




Synthesis and stability study of a new major metabolite of γ-hydroxybutyric acid
Author(s): Ida Nymann Petersen | Jesper Langgaard Kristensen | Christian Tortzen | Torben Breindahl | Daniel Sejer Pedersen
Volume: 9
Issue: 1
Year: 2013




Regio- and stereoselective carbometallation reactions of N-alkynylamides and sulfonamides
Author(s): Yury Minko | Morgane Pasco | Helena Chechik | Ilan Marek
Volume: 9
Issue: 1
Year: 2013




Metal-mediated aminocatalysis provides mild conditions: Enantioselective Michael addition mediated by primary amino catalysts and alkali-metal ions
Author(s): Matthias Leven | Jörg M. Neudörfl | Bernd Goldfuss
Volume: 9
Issue: 1
Year: 2013




Chemoenzymatic synthesis and biological evaluation of enantiomerically enriched 1-(β-hydroxypropyl)imidazolium- and triazolium-based ionic liquids
Author(s): Paweł Borowiecki | Małgorzata Milner-Krawczyk | Jan Plenkiewicz
Volume: 9
Issue: 1
Year: 2013




Electron and hydrogen self-exchange of free radicals of sterically hindered tertiary aliphatic amines investigated by photo-CIDNP
Author(s): Martin Goez | Isabell Frisch | Ingo Sartorius
Volume: 9
Issue: 1
Year: 2013




The β-cyclodextrin/benzene complex and its hydrogen bonds – a theoretical study using molecular dynamics, quantum mechanics and COSMO-RS
Author(s): Jutta Erika Helga Köhler | Nicole Grczelschak-Mick
Volume: 9
Issue: 1
Year: 2013




Easy and direct conversion of tosylates and mesylates into nitroalkanes
Author(s): Alessandro Palmieri | Serena Gabrielli | Roberto Ballini
Volume: 9
Issue: 1
Year: 2013




Presence or absence of a novel charge-transfer complex in the base-catalyzed hydrolysis of N-ethylbenzamide or ethyl benzoate
Author(s): Shinichi Yamabe | Wei Guan | Shigeyoshi Sakaki
Volume: 9
Issue: 1
Year: 2013




Synthesis of 2,3-dihydronaphtho[2,3-d][1,3]thiazole-4,9-diones and 2,3-dihydroanthra[2,3-d][1,3]thiazole-4,11-diones and novel ring contraction and fusion reaction of 3H-spiro[1,3-thiazole-2,1'-cyclohexanes] into 2,3,4,5-tetrahydro-1H-carbazole-6,11-diones
Author(s): Lidia S. Konstantinova | Kirill A. Lysov | Ljudmila I. Souvorova | Oleg A. Rakitin
Volume: 9
Issue: 1
Year: 2013




Glycosylation efficiencies on different solid supports using a hydrogenolysis-labile linker
Author(s): Mayeul Collot | Steffen Eller | Markus Weishaupt | Peter H. Seeberger
Volume: 9
Issue: 1
Year: 2013




Efficient synthesis of phenylene-ethynylene rods and their use as rigid spacers in divalent inhibitors
Author(s): Francesca Pertici | Norbert Varga | Arnoud van Duijn | Matias Rey-Carrizo | Anna Bernardi | Roland J. Pieters
Volume: 9
Issue: 1
Year: 2013



